Система малярийный паразит — эритроцит: биохимические основы и действие антималярийных препаратов
Диссертация
Переходя к проблемам лекарственного воздействия на пораженный эритроцит, следует отметить, что биохимические реакции, лежащие в основе терапевтического действия многих современных антималярийных препаратов, остаются неизвестными. В первую очередь, это относится к многочисленным соединениям хинолино-вого ряда, обладающим шизонтоцидной активностью в отношении кровяных форм малярийных паразитов… Читать ещё >
Содержание
- ОБЩАЯ ХАРАКТЕРИСТИКА. РАБОТЫ
- ГЛАВА I. СИСТЕМА КРАСНОЙ КРОВИ ПРИ МАЛЯРИИ
- ЭКСПЕРИМЕНТАЛЬНЫЕ МОДЕЛИ И ПРЕПАРАТИВНЫЕ МЕТОДЫ ИССЛЕДОВАНИЙ
- I. I* Обзор литературы
- 1. 1. 1. Краткая характеристика возбудителя
- 1. 1. 2. Некоторые гематологические аспекты малярии
- 1. 1. 3. Препаративные методы исследований эритро-цитарных форм малярийных паразитов
- 1. 2. Экспериментальная часть
- 1. 2. 1. Паразитешя и возрастные цопуляции эритроцитов у крыс, зараженных Plasmodium berghe
- 1. 2. 2. Паразитологическая и гематологическая характеристика мышей, зараженных p. berghe
- 1. 2. 3. Удаление лейкоцитов, отделение пораженных эритроцитов, возрастное фракционирование паразитов
- 1. 3. Резюме
- I. I* Обзор литературы
- 2. 1. " Физико-химические параметры транспорта газов и буферной емкости крови
- 2. 2. История изучения кислородного и кислотно-щелочного баланса крови при малярии
- 2. 3. Кислородный баланс крови при экспериментальной малярии, ВЫЗВаННОЙ P. berghe
- 2. 4. Кислотно-щелочное равновесие крови при экспериментальной маЛЯрИИ, ВЫЗВаННОЙ P. berghe
- 2. 5. Влияние внутриклеточного паразита на функцию гемоглобина
- 2. 6. Резюме
- 3. 1. Обзор литературы
- 3. 1. 1. Энергетика и гликолиз
- 3. 1. 2. Система глутатиона и пентозо-фосфатный
- 3. 1. 3. Антиоксидантная система и другие реакции НО
- 3. 2. Собственные исследования
- 3. 2. 1. Энергетическая характеристика эритроцитов при малярийной инфекции, вызванной
- F. berghe
- 3. 2. 2. Гликолиз в эритроцитах, пораженных
- P. berghe
- 3. 2. 3. Восстановленный глутатион в пораженных эритроцитах
- 3. 2. 4. Гемоглобин и аспартатаминотрансфераза в пораженных эритроцитах
- 3. 2. 5. Ферменты пентозо-фосфатного пути в пораженных эритроцитах
- 3. 2. 6. Ферментативная защита клетки от окисления
- 3. 2. 7. Ферментативное окисление пиридиннуклеотидов в метаболизме эритроцита и паразита
- 3. 3. Интеграция и регуляция метаболизма в системе паразит-эритроцит
- 3. 4. Резюме
- 4. 1. Обзор литературы
- 4. 1. 1. Биохимические механизмы шизонтоцидного действия аминохинолинов.. ¦
- 4. 1. 2. Биохимические механизмы гемолитического действия 8-аминохинолинов
- 4. 2. Экспериментальное изучение антималярийного действия соединений ряда хинолина
- 4. 2. 1. Гликолиз в пораженных эритроцитах под действием антималярийных соединений
- 4. 2. 2. Взаимодействие аминохинолинов с феррите
- 4. 2. 3. Дополнительные исследования механизмов антималярийной активности производных хинолина
- 4. 3. Экспериментальное изучение гемолитического действия примахина
- 4. 3. 1. Модель для изучения гемолиза in vitro
- 4. 3. 2. Роль супероксида в окислительном повреждении эритроцитов примахином
- 4. 3. 3. Защитный эффект антиоксидантов в отношении гемолиза, индуцированного примахином
- 4. 4. Резюме
- 5. 1. Биохимические основы взаимодействия малярийного паразита с эритроцитом хозяина
- 5. 2. Использование полученных результатов в научных исследованиях, диагностике и лечении малярии
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